SCHEMBL29133055

SCHEMBL29133055

COCc1cc(-c2nnc(C3CC3)o2)ccc1Br

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.52
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
KDM4E B2RXH2 1/20 0.43
MAPT P10636 5/20 0.42
MAPK1 P28482 1/20 0.42
ALOX15B O15296 1/20 0.42
POLB P06746 1/20 0.40
CYP2C19 P33261 1/20 0.40
LRRK2 Q5S007 1/20 0.40
TP53 P04637 2/20 0.39
TLR9 Q9NR96 3/20 0.39
TLR8 Q9NR97 3/20 0.39
TLR7 Q9NYK1 3/20 0.39
PIM1 P11309 2/20 0.38
PIM2 Q9P1W9 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29132973 0.85 ALDH1A1 (0.38) ALDH1A1CA1CA2KDM4EMAPT
SCHEMBL29133063 0.81 ALDH1A1 (0.52) ALDH1A1CA1CA2KDM4EMAPT
SCHEMBL29133160 0.80 SMN1; SMN2 (0.41) ALDH1A1KDM4EMAPTMAPK1POLB
SCHEMBL29133064 0.80 NOTUM (0.43) ALDH1A1KDM4EMAPTMAPK1POLB
SCHEMBL29133017 0.79 DGAT1 (0.50) ALDH1A1KDM4EMAPTMAPK1POLB
SCHEMBL29133128 0.78 ALDH1A1 (0.39) ALDH1A1CA1CA2MAPTLRRK2
SCHEMBL30622248 0.78 KDM4E (0.49) ALDH1A1CA1CA2KDM4EMAPT
SCHEMBL29133117 0.76 HDAC6 (0.45)
SCHEMBL30622235 0.75 ALDH1A1 (0.52) ALDH1A1CA1CA2KDM4EMAPT
SCHEMBL29133060 0.75 ALDH1A1 (0.43) ALDH1A1CA1CA2KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed