SCHEMBL29133048

SCHEMBL29133048

COCc1c(Br)ccc(-c2nnc(C3CC3)o2)c1F

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
LRRK2 Q5S007 1/20 0.36
TP53 P04637 4/20 0.35
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34
HTR4 Q13639 5/20 0.34
FLT3 P36888 2/20 0.34
CYP2C19 P33261 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29133128 0.76 ALDH1A1 (0.39) ALDH1A1CA1CA2LRRK2TP53
SCHEMBL29133055 0.73 ALDH1A1 (0.52) ALDH1A1CA1CA2LRRK2TP53
SCHEMBL29133060 0.73 ALDH1A1 (0.43) ALDH1A1CA1CA2LRRK2MAPT
SCHEMBL30622258 0.73 ALDH1A1 (0.43) ALDH1A1CA1CA2LRRK2MAPT
SCHEMBL29133171 0.70 TP53 (0.42) ALDH1A1CA1CA2LRRK2TP53
SCHEMBL30622188 0.69 ALDH1A1 (0.39) ALDH1A1CA1CA2LRRK2TP53
SCHEMBL29133172 0.69 ALDH1A1 (0.39) ALDH1A1CA1CA2LRRK2TP53
SCHEMBL29133061 0.69 TP53 (0.45) ALDH1A1CA1CA2LRRK2TP53
SCHEMBL29133063 0.69 ALDH1A1 (0.52) ALDH1A1CA1CA2LRRK2MAPT
SCHEMBL24725043 0.65 ADRA1A (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed