SCHEMBL29133060

SCHEMBL29133060

COCc1nc(-c2nnc(C3CC3)o2)ccc1Br

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
SMO Q99835 1/20 0.37
MAPT P10636 2/20 0.36
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALOX15B O15296 1/20 0.34
APLNR P35414 1/20 0.34
HTR4 Q13639 5/20 0.33
FLT3 P36888 1/20 0.33
LRRK2 Q5S007 1/20 0.33
ATR Q13535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30622258 1.00 ALDH1A1 (0.43) ALDH1A1CA1CA2SMOMAPT
SCHEMBL30622257 0.81 BRD4 (0.36) GAA
SCHEMBL29133136 0.80 TDP1 (0.36) ALDH1A1MAPTKDM4ENPC1RAB9A
SCHEMBL30622228 0.80 TDP1 (0.36) ALDH1A1MAPTKDM4ENPC1RAB9A
SCHEMBL29133005 0.76 HDAC6 (0.39)
SCHEMBL30622220 0.76 HDAC6 (0.39)
SCHEMBL29133055 0.75 ALDH1A1 (0.52) ALDH1A1CA1CA2MAPTKDM4E
SCHEMBL29133048 0.73 ALDH1A1 (0.42) ALDH1A1CA1CA2MAPTMAPK1
SCHEMBL29133063 0.68 ALDH1A1 (0.52) ALDH1A1CA1CA2MAPTKDM4E
SCHEMBL24921754 0.67 BRD4 (0.38) MAPTNPC1RAB9AL3MBTL1ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088884-A Imidazopyridazine derivatives as GABAA receptor modulators, pharmaceutical compositions and uses 上海赛默罗德生物科技有限公司 2023-11-21 CN disclosed