SCHEMBL29134294

SCHEMBL29134294

N#CC(CCO)(CCO)c1ccc(Br)cc1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.35
HSD17B10 Q99714 1/20 0.35
RECQL P46063 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
CYP2A6 P11509 1/20 0.31
OGG1 O15527 1/20 0.31
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16136803 0.80 DRD2 (0.42)
SCHEMBL11091213 0.79 ALDH1A1 (0.40) HSD17B10RECQLESR1ESR2OGG1
SCHEMBL5469510 0.77 HSD17B10 (0.45) CASP1HSD17B10RECQLALOX15
SCHEMBL1141384 0.76 CA1 (0.34) CASP1HSD17B10ESR1ESR2CYP2A6
SCHEMBL29134450 0.75 CA1 (0.33) CASP1HSD17B10
SCHEMBL9451781 0.72 CA1 (0.32) CASP1HSD17B10
SCHEMBL15774978 0.69 ESR1 (0.47) RECQLESR1ESR2CYP2A6OGG1
SCHEMBL5476420 0.68 KCNN4 (0.41) CASP1HSD17B10
SCHEMBL5476864 0.68 CTSK (0.41)
SCHEMBL31634536 0.67 KMT2A (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed