SCHEMBL29134300

SCHEMBL29134300

CS(=O)(=O)NC1CS(=O)(=O)c2cc(Br)ccc21

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 2/20 0.33
SLC22A12 Q96S37 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1530500 0.74 GRIA2 (0.44) CA1CA2CA9
SCHEMBL22439483 0.71 TGM2 (0.40)
SCHEMBL24698411 0.71 AAK1 (0.38)
SCHEMBL30015258 0.71 AAK1 (0.38)
SCHEMBL2589648 0.70 VEGFA (0.39) CA1CA2CA9
SCHEMBL22438912 0.70 KDM1A (0.39) CA1CA2CA9
SCHEMBL29134322 0.68 ADRA2A (0.42) CA2
SCHEMBL29134339 0.67 SRD5A1 (0.32) SLC22A12
SCHEMBL30014797 0.67 SRD5A1 (0.32) SLC22A12
SCHEMBL8160279 0.65 GRIA2 (0.44) CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed