SCHEMBL29134322

SCHEMBL29134322

CS(=O)(=O)NC1CCOc2cc(Br)ccc21

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.42
KDM4C Q9H3R0 1/20 0.39
HTR2A P28223 3/20 0.38
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
HTT P42858 1/20 0.37
BLM P54132 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
CA2 P00918 1/20 0.34
HSD17B2 P37059 1/20 0.34
ALDH1A1 P00352 1/20 0.33
HTR6 P50406 1/20 0.33
MAP3K14 Q99558 1/20 0.33
PKM P14618 1/20 0.33
PKLR P30613 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24698005 0.89 ADRA2A (0.42) ADRA2AKDM4CHTR2ADRD2DRD3
SCHEMBL28449906 0.81 ADRA2A (0.47) ADRA2AKDM4CHTR2ALMNAMAPT
SCHEMBL16794282 0.76 KDM4C (0.47) ADRA2AKDM4CTRPV1HSD17B2MAOB
SCHEMBL23976524 0.76 KDM4C (0.42) ADRA2AKDM4CHTR2ATRPV1HSD17B2
SCHEMBL1530500 0.75 GRIA2 (0.44) TRPV1CA2MAOB
SCHEMBL6337557 0.72 DRD2 (0.42) HTR2ADRD2DRD3HTTCA2
SCHEMBL19889279 0.72 ADRA2A (0.50) ADRA2AKDM4CHTR2ALMNAMAPT
SCHEMBL27898816 0.72 ALDH1A1 (0.46) ADRA2AKDM4CALDH1A1
SCHEMBL16814170 0.72 AAK1 (0.41) ADRA2AKDM4CTRPV1HSD17B2
SCHEMBL15897694 0.69 KDM4C (0.43) ADRA2AKDM4CLMNAMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed