SCHEMBL29134754

SCHEMBL29134754

CC1(C)OB(c2ccc3[nH]c(C(N)=O)cc3c2)OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.40
MMP13 P45452 1/20 0.40
F11 P03951 3/20 0.40
F2 P00734 2/20 0.40
PRSS1 P07477 2/20 0.40
PRSS2 P07478 2/20 0.40
PRSS3 P35030 2/20 0.40
PIN1 Q13526 1/20 0.39
PDGFRB P09619 3/20 0.38
FLT3 P36888 3/20 0.38
ABL1 P00519 1/20 0.38
KIT P10721 1/20 0.38
BCR P11274 1/20 0.38
P4HB P07237 1/20 0.38
CYP2D6 P10635 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
PDGFRA P16234 2/20 0.38
CFD P00746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13830366 0.88 PIN1 (0.54) PIN1PDGFRBFLT3ABL1KIT
SCHEMBL2735974 0.84 XDH (0.50) MMP2MMP13PIN1PDGFRBFLT3
SCHEMBL488403 0.81 KDM4E (0.61) MMP2MMP13CYP2D6SLC6A2SLC6A4
SCHEMBL31692446 0.78 PYGL (0.43) PIN1PDGFRBP4HBCYP2D6SLC6A2
SCHEMBL3190570 0.77 CYP2A6 (0.46) F11CA1CA2CA9LPL
SCHEMBL20611918 0.77 EIF4A3 (0.50) F11F2PRSS1PRSS2PRSS3
SCHEMBL15642715 0.75 NPC1 (0.48) KDM4EALDH1A1LMNAHPGD
SCHEMBL28292828 0.75 CYP2A6 (0.45) F11P4HBCA1CA2CA9
SCHEMBL2098959 0.74 CA9 (0.50) F11CA1CA2CA9LPL
SCHEMBL16567346 0.74 LPL (0.42) F11F2PRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed