SCHEMBL29134875

SCHEMBL29134875

CC(C)(C)OC(=O)NCC(F)(F)c1ccc(Br)cc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.46
RECQL P46063 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
FPR3 P25089 6/20 0.44
FPR2 P25090 6/20 0.44
CTSS P25774 2/20 0.43
CTSK P43235 2/20 0.43
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
AAK1 Q2M2I8 4/20 0.40
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
IDO1 P14902 1/20 0.38
CTSB P07858 1/20 0.37
AKT1 P31749 1/20 0.37
APLNR P35414 1/20 0.37
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24891906 0.85 EPHX2 (0.40) LMNAPOLBIDO1
SCHEMBL28294256 0.83 CTSB (0.47) SMN1; SMN2CTSSCTSKLMNAPOLB
SCHEMBL21437078 0.82 STK17B (0.38) FPR3FPR2LMNAPOLBIDO1
SCHEMBL24891861 0.81 ALDH1A1 (0.46) NPC1RAB9ASMN1; SMN2LMNAPOLB
SCHEMBL13262888 0.80 AAK1 (0.46) NPC1RECQLRAB9ASMN1; SMN2FPR3
SCHEMBL15739717 0.77 NPC1 (0.46) NPC1RECQLRAB9ASMN1; SMN2FPR3
SCHEMBL81094 0.75 FPR3 (0.58) NPC1RECQLRAB9ASMN1; SMN2FPR3
SCHEMBL31306453 0.75 GSK3B (0.39) RECQLMAPT
SCHEMBL4901469 0.75 FPR3 (0.55) NPC1RECQLRAB9ASMN1; SMN2FPR3
SCHEMBL28654685 0.74 LMNA (0.41) NPC1RAB9ASMN1; SMN2FPR3FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4313967-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2024-02-07 EP disclosed
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed
WO-2022212194-A1 KHK INHIBITORS GILEAD SCIENCES, INC. (US) 2022-10-06 WO disclosed