SCHEMBL29134937

SCHEMBL29134937

COc1cc(NS(=O)(=O)c2cc(Br)ccc2OC)ccc1C#N

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 1/20 0.58
TRIM24 O15164 1/20 0.57
ALPL P05186 6/20 0.56
SHMT2 P34897 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
KMT2A Q03164 2/20 0.54
MEN1 O00255 1/20 0.54
BRD4 O60885 2/20 0.53
BRD2 P25440 1/20 0.53
GLA P06280 1/20 0.52
WDR5 P61964 2/20 0.49
EDNRB P24530 2/20 0.49
EDNRA P25101 2/20 0.49
KDM4E B2RXH2 1/20 0.49
GAA P10253 1/20 0.49
PKM P14618 1/20 0.49
MYC P01106 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29134425 0.90 SLC22A12 (0.73) SLC22A12TRIM24ALPLSHMT2SMN1; SMN2
SCHEMBL29134947 0.85 ALPL (0.58) TRIM24ALPLSMN1; SMN2KMT2AMEN1
SCHEMBL18530464 0.79 ALPL (0.70) ALPLSMN1; SMN2KMT2AMEN1GLA
SCHEMBL21761109 0.78 LMNA (0.73) ALPLSMN1; SMN2KMT2AMEN1GLA
SCHEMBL21760616 0.78 ALPL (0.62) TRIM24ALPLSMN1; SMN2KMT2AMEN1
SCHEMBL3761698 0.78 ALPL (0.72) ALPLSMN1; SMN2KMT2AMEN1GLA
SCHEMBL14018775 0.76 ALPL (0.59) ALPLSMN1; SMN2KMT2ABRD4BRD2
SCHEMBL329987 0.76 TP53 (0.73) ALPLSMN1; SMN2KMT2AGLAWDR5
SCHEMBL21761107 0.75 ALPL (0.65) ALPLSMN1; SMN2KMT2AMEN1BRD4
SCHEMBL286644 0.75 AR (0.53) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117120429-A KHK inhibitor 吉利德科学公司 2023-11-24 CN disclosed