Thiophene Carboxylic Acid

Thiophene Carboxylic Acid

SCHEMBL29135076

NC(=O)c1cccc(S(=O)(=O)N2CCc3ccccc3C2)c1.O=C(O)c1cccs1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 17/20 0.77
AKR1C1 Q04828 4/20 0.68
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
PPARG P37231 1/20 0.56
PPARD Q03181 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
MAPT P10636 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2011206 0.82 AKR1C3 (1.00) AKR1C3AKR1C1MEN1KMT2AALDH1A1
SCHEMBL30819658 0.82 AKR1C3 (1.00) AKR1C3AKR1C1MEN1KMT2AALDH1A1
Thiophene Carboxylic Acid SCHEMBL29135074 0.81 AKR1C3 (0.70) AKR1C3AKR1C1MEN1KMT2AALDH1A1
SCHEMBL14943437 0.76 AKR1C3 (0.79) AKR1C3AKR1C1MEN1KMT2APPARG
Carbamic Acid SCHEMBL27693825 0.75 AKR1C3 (0.60) AKR1C3AKR1C1MEN1KMT2AALDH1A1
SCHEMBL23081190 0.75 AKR1C3 (0.78) AKR1C3AKR1C1MEN1KMT2AALDH1A1
SCHEMBL12401136 0.73 AKR1C3 (0.74) AKR1C3AKR1C1MEN1KMT2APPARG
SCHEMBL21067755 0.72 PPARG (1.00) AKR1C3AKR1C1MEN1KMT2APPARG
SCHEMBL29134720 0.72 NR3C1 (0.61) AKR1C3AKR1C1ALDH1A1LMNAMAPT
SCHEMBL693455 0.71 KMT2A (1.00) AKR1C3AKR1C1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117298108-A Androgen receptor and glucocorticoid receptor dual-target inhibitor and application thereof 浙江师范大学 2023-12-29 CN disclosed