SCHEMBL29137977

SCHEMBL29137977

C=Cc1cccc2cnc(OC(N)=O)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.39
SLC9A1 P19634 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PIM1 P11309 1/20 0.33
PSMD14 O00487 1/20 0.33
STAMBP O95630 1/20 0.33
COPS5 Q92905 1/20 0.33
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PLK4 O00444 1/20 0.30
CHEK1 O14757 1/20 0.30
AURKA O14965 1/20 0.30
DAPK3 O43293 1/20 0.30
MAP4K4 O95819 1/20 0.30
CSF1R P07333 1/20 0.30
RET P07949 1/20 0.30
FGFR1 P11362 1/20 0.30
PDGFRA P16234 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29137983 0.88 MEN1 (0.37) PARP1MEN1KMT2APIM1PSMD14
SCHEMBL4073461 0.75 PLAU (0.46) PARP1MEN1KMT2APSMD14STAMBP
SCHEMBL30636265 0.75 PLAU (0.46) PARP1MEN1KMT2APSMD14STAMBP
SCHEMBL29137986 0.74
SCHEMBL2145623 0.70 CYP1A2 (0.48) PARP1MEN1KMT2APSMD14COPS5
SCHEMBL26933015 0.70 ALDH1A1 (0.38) PARP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL29890165 0.70 ALDH1A1 (0.38) PARP1MEN1KMT2AKDM4EALDH1A1
SCHEMBL29137974 0.69 ERN1 (0.34)
SCHEMBL4020792 0.68 LMNA (0.39) MEN1KMT2AKDM4EALDH1A1HSD17B10
SCHEMBL28849760 0.67 PARP1 (0.40) PARP1MEN1KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117062804-A 1, 3-substituted cyclobutyl derivatives and their use 诺华股份有限公司 2023-11-14 CN disclosed