SCHEMBL29139949

SCHEMBL29139949

Brc1ccc(C2CCCN2c2ccccc2C2CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.43
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
NUDT1 P36639 2/20 0.40
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP2C19 P33261 1/20 0.39
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24775204 0.81 NOS1 (0.44) NOS1KDM4EALDH1A1GAAMAPT
SCHEMBL28528279 0.77 CYP2D6 (0.38) NOS1CYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL28528284 0.77 CYP2D6 (0.38) NOS1CYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL22165467 0.74 CHRNB2 (0.50) NUDT1CYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL28519576 0.73 NOS1 (0.37) NOS1KDM4EALDH1A1GAAMAPT
SCHEMBL24775580 0.72 HRH3 (0.38) MAPTCYP2D6CYP2C9MAPK1CYP2C19
SCHEMBL28522996 0.72 HDAC1 (0.40)
SCHEMBL6937201 0.72 NOS1 (0.40) NOS1KDM4EALDH1A1GAAMAPT
SCHEMBL24775532 0.71 MGLL (0.41) NOS1KDM4EALDH1A1GAAMAPT
SCHEMBL29855684 0.71 MGLL (0.41) NOS1KDM4EALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117683029-A Bcl-2 inhibitors 百济神州有限公司 2024-03-12 CN disclosed
CN-117430601-A Bcl-2 inhibitors 百济神州有限公司 2024-01-23 CN disclosed
CN-112437772-B Bcl-2 inhibitors 百济神州有限公司 2023-11-21 CN disclosed