SCHEMBL29149786

SCHEMBL29149786

COC(=O)c1ccc2nc(C=C3CCN(C(=O)OC(C)(C)C)CC3)n(C[C@@H]3CCO3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.39
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
ACSS2 Q9NR19 2/20 0.37
GPR119 Q8TDV5 7/20 0.37
GRM5 P41594 1/20 0.37
MAPT P10636 3/20 0.36
SCN9A Q15858 1/20 0.36
TP53 P04637 1/20 0.36
THRB P10828 1/20 0.36
HDAC4 P56524 1/20 0.35
BRD4 O60885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29149793 1.00 PKM (0.39) PKMALDH1A1MAPK1ACSS2GPR119
SCHEMBL30680670 1.00 PKM (0.39) PKMALDH1A1MAPK1ACSS2GPR119
SCHEMBL30680774 1.00 PKM (0.39) PKMALDH1A1MAPK1ACSS2GPR119
SCHEMBL29149806 0.92 GLP1R (0.40)
SCHEMBL29149813 0.92 GLP1R (0.40)
SCHEMBL29924743 0.92 GLP1R (0.40)
SCHEMBL30680745 0.84 ALDH1A1 (0.41) ALDH1A1MAPK1ACSS2MAPT
SCHEMBL29150155 0.84 ALDH1A1 (0.41) ALDH1A1MAPK1ACSS2MAPT
SCHEMBL29150154 0.84 ALDH1A1 (0.41) ALDH1A1MAPK1ACSS2MAPT
SCHEMBL24266522 0.82 RORC (0.46) PKMALDH1A1MAPK1ACSS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117177970-A Polycyclic derivative regulator, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-12-05 CN disclosed
WO-2022228490-A1 POLYCYCLIC DERIVATIVE MODULATOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF 上海翰森生物医药科技有限公司 2022-11-03 WO disclosed