SCHEMBL29167207

SCHEMBL29167207

Nc1nc(N)nc(NCC2CCOCC2)n1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH3 Q9ULD8 1/20 0.54
ALDH1A1 P00352 1/20 0.42
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
HRH4 Q9H3N8 3/20 0.40
DHFR P00374 1/20 0.39
DCPS Q96C86 1/20 0.39
TPH1 P17752 1/20 0.38
RIPK2 O43353 1/20 0.37
APP P05067 1/20 0.36
CSF1R P07333 1/20 0.36
VNN1 O95497 1/20 0.36
KCNH2 Q12809 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
HIF1A Q16665 1/20 0.34
JAK2 O60674 1/20 0.34
JAK3 P52333 1/20 0.34
CHUK O15111 1/20 0.34
CCNK O75909 1/20 0.34
CDK9 P50750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8053409 0.81 APP (0.51) PTGS2HRH4TPH1APPKCNH2
SCHEMBL29197980 0.79 KCNH3 (0.54) KCNH3ALDH1A1PTGS1PTGS2RIPK2
SCHEMBL8039831 0.78 APP (0.51) KCNH3PTGS2HRH4TPH1APP
SCHEMBL23175130 0.77 HRH4 (0.54) HRH4KCNH2HRH3
SCHEMBL30784995 0.72 MAPK1 (0.53) PTGS2HRH4KCNH2
SCHEMBL15668792 0.72 ALDH1A1 (0.37) KCNH3ALDH1A1HRH4
SCHEMBL29197978 0.72 HRH4 (0.42) KCNH3ALDH1A1HRH4DHFRDCPS
SCHEMBL9912549 0.70 KCNH3 (0.49) KCNH3ALDH1A1PTGS1PTGS2RIPK2
SCHEMBL16094915 0.70 NPY5R (0.40) KCNH3ALDH1A1HRH4TPH1APP
SCHEMBL31229795 0.69 KCNH3 (0.45) KCNH3ALDH1A1PTGS1PTGS2RIPK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117624137-A Triazine skeleton small molecule heparin reversal agent and preparation method and application thereof 中国药科大学 2024-03-01 CN disclosed
CN-117417328-A Triazine compound for reversing anticoagulant activity of low-molecular heparin, and preparation method and application thereof 中国药科大学 2024-01-19 CN disclosed