SCHEMBL29174264

SCHEMBL29174264

COC(=O)Cc1cc(Cl)ccc1-c1nnn[nH]1.COC(=O)Cc1cc(Cl)ccc1C#N

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.35
HPGD P15428 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
KLKB1 P03952 1/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
NOS3 P29474 4/20 0.34
NOS1 P29475 4/20 0.34
NOS2 P35228 4/20 0.34
S1PR3 Q99500 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
F2 P00734 1/20 0.34
ALPL P05186 1/20 0.33
XDH P47989 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27033945 0.90 ALPL (0.38) KDM4EMAPTGAAALPLMEN1
SCHEMBL27033421 0.82 MAPT (0.46) ADRA1DHPGDNPSR1KDM4EMAPT
SCHEMBL29958664 0.82 MAPT (0.46) ADRA1DHPGDNPSR1KDM4EMAPT
SCHEMBL3834764 0.79 EGFR (0.43) KDM4EMAPTGAAALPL
SCHEMBL29958529 0.76 KEAP1 (0.40) KDM4EMAPTCYP2C9ALPLALDH1A1
SCHEMBL27033835 0.76 KEAP1 (0.40) KDM4EMAPTCYP2C9ALPLALDH1A1
SCHEMBL6816520 0.74 PRMT5 (0.36) HPGDKDM4EMAPTGAATDP1
SCHEMBL29174287 0.74 MEN1 (0.33) HPGDKDM4EMAPTGAATDP1
SCHEMBL28068640 0.72 HPGD (0.45) HPGDNPSR1KDM4EMAPTCYP1A2
SCHEMBL1307875 0.70 GAA (0.53) KDM4EMAPTCYP1A2CYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396474-A Plasma kallikrein inhibitors 武田药品工业株式会社 2024-01-12 CN disclosed