SCHEMBL29178282

SCHEMBL29178282

COc1ccnc(NC(=O)N2CCN(c3ccccc3)CC2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 6/20 0.60
KMT2A Q03164 3/20 0.56
GAA P10253 1/20 0.56
NOS3 P29474 1/20 0.54
NOS1 P29475 1/20 0.54
NOS2 P35228 1/20 0.54
ALDH1A1 P00352 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
RBP4 P02753 1/20 0.54
MAPT P10636 3/20 0.53
MAPK1 P28482 2/20 0.53
MEN1 O00255 1/20 0.53
HCRTR1 O43613 1/20 0.53
USP2 O75604 1/20 0.53
CYP1A2 P05177 1/20 0.53
POLB P06746 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13234915 0.78 MAPT (0.77) KMT2AGAAALDH1A1SMN1; SMN2MAPT
SCHEMBL6966880 0.77 FAAH (0.55) KMT2AGAAALDH1A1SMN1; SMN2MAPT
SCHEMBL6956624 0.76 NPY5R (0.58) KMT2AALDH1A1SMN1; SMN2MAPTMAPK1
SCHEMBL8699365 0.75 ALDH1A1 (0.58) KMT2AGAAALDH1A1RBP4MAPT
SCHEMBL20072349 0.75 PHGDH (0.77) PHGDHKMT2AGAANOS3NOS1
SCHEMBL20063159 0.75 PHGDH (1.00) PHGDH
SCHEMBL13996934 0.74 MET (0.57) PHGDHNOS3NOS1NOS2POLB
SCHEMBL4916560 0.74 HTT (0.52) KMT2AGAAALDH1A1SMN1; SMN2RBP4
SCHEMBL1138338 0.74 HTT (0.52) KMT2AGAAALDH1A1SMN1; SMN2RBP4
SCHEMBL25189182 0.74 RIOK2 (0.60) PHGDHNOS3NOS1NOS2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117736163-A Phenylpiperazine derivative or pharmaceutical salt thereof, preparation method and application thereof in preparation of pain treatment drugs 郑州大学第一附属医院 2024-03-22 CN claimed
CN-117736163-A Phenylpiperazine derivative or pharmaceutical salt thereof, preparation method and application thereof in preparation of pain treatment drugs 郑州大学第一附属医院 2024-03-22 CN disclosed