SCHEMBL291859

SCHEMBL291859

C=C[C@H](COCc1ccccc1)OC(=O)CC(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.42
CA2 P00918 2/20 0.42
CA7 P43166 2/20 0.42
CA9 Q16790 2/20 0.42
KMT2A Q03164 1/20 0.41
HTT P42858 1/20 0.40
TSHR P16473 1/20 0.40
SLC1A1 P43005 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
NPC1 O15118 1/20 0.40
FAAH O00519 3/20 0.39
MAPK1 P28482 1/20 0.39
MMP9 P14780 1/20 0.38
MMP14 P50281 1/20 0.38
PSMB11 A5LHX3 1/20 0.38
PSMD11 O00231 1/20 0.38
PSMD12 O00232 1/20 0.38
PSMD14 O00487 1/20 0.38
PSMA7 O14818 1/20 0.38
PSMD3 O43242 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL291860 1.00 CA1 (0.42) CA1CA2CA7CA9KMT2A
SCHEMBL2074009 0.83 ALDH1A1 (0.47) CA1CA2CA7CA9KMT2A
SCHEMBL6337071 0.81 CA1 (0.46) CA1CA2CA7CA9KMT2A
SCHEMBL6337069 0.81 CA1 (0.46) CA1CA2CA7CA9KMT2A
SCHEMBL9489310 0.75 HTT (0.49) CA1CA2CA7CA9KMT2A
SCHEMBL9489307 0.75 HTT (0.49) CA1CA2CA7CA9KMT2A
SCHEMBL9489505 0.75 HTT (0.49) CA1CA2CA7CA9KMT2A
SCHEMBL7596298 0.75 PRKCA (0.45) TSHRMMP9
SCHEMBL8419725 0.75 CA1 (0.51) CA1CA2CA7CA9KMT2A
SCHEMBL22918182 0.74 KMT2A (0.56) CA1CA2CA7CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158790-B2 Cyclic amine compound DAIICHI SANKYO COMPANY, LIMITED (JP) 2012-04-17 US disclosed
EP-2036896-B1 CYCLIC AMINE COMPOUND DAIICHI SANKYO CO LTD (JP) 2012-03-14 EP disclosed