SCHEMBL2918657

SCHEMBL2918657

CCOC(=O)Oc1cc(Cl)ncn1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CUL4A Q13619 2/20 0.38
KMT2A Q03164 2/20 0.37
RAB9A P51151 1/20 0.37
SOAT1 P35610 1/20 0.36
DGAT1 O75907 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
KDR P35968 1/20 0.34
CA2 P00918 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1934857 0.81 L3MBTL1 (0.37) JAK2ALDH1A1CUL4AKMT2ASMN1; SMN2
SCHEMBL27820544 0.77 KDM4E (0.38) ALDH1A1KMT2ARAB9ASMN1; SMN2TSHR
SCHEMBL11697983 0.77 ALOX15 (0.38) ALDH1A1KMT2ARAB9AKDRCA2
SCHEMBL9101158 0.76 CUL4A (0.40) JAK2JAK1TYK2JAK3ALDH1A1
SCHEMBL14387902 0.76 ALDH1A1 (0.39) ALDH1A1KMT2ARAB9A
SCHEMBL9326634 0.75 JAK2 (0.46) JAK2JAK1TYK2JAK3ALDH1A1
SCHEMBL549184 0.75 CYP1A2 (0.47) ALDH1A1KMT2ARAB9ACYP2C9CYP2C19
SCHEMBL1742128 0.74 KMO (0.35) KMT2A
SCHEMBL3660791 0.74 KMO (0.38) KMT2A
SCHEMBL3997981 0.74 CUL4A (0.48) JAK2JAK1TYK2JAK3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225223-B1 ORGANIC COMPOUNDS BOEHRINGER INGELHEIM INT (DE) 2017-01-11 EP disclosed
EP-2225227-B1 1',3'-Dihydrospiro[imidazolidin-4,2'-inden]-2,5-diones and 1,3-dihydrospiro[inden-2,3']-pyrroles as CGRP antagonists BOEHRINGER INGELHEIM INT (DE) 2015-08-26 EP disclosed
EP-2251339-A2 COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed
EP-2251338-A2 Organic compounds Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed
EP-2225223-A2 ORGANIC COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
EP-2225227-A2 COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
WO-2009065920-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed
WO-2009065919-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed
EP-2062889-A1 Compounds Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-05-27 EP disclosed