SCHEMBL29201269

SCHEMBL29201269

O=C(CBr)C1(c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.51
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
TSHR P16473 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP2C19 P33261 2/20 0.48
LMNA P02545 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
ALOX15 P16050 1/20 0.48
NPSR1 Q6W5P4 2/20 0.46
MAPT P10636 1/20 0.46
HTR1E P28566 1/20 0.46
S1PR3 Q99500 1/20 0.46
CYP2C9 P11712 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CES1 P23141 1/20 0.42
HDAC1 Q13547 1/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1769201 0.80 NPSR1 (0.50) MEN1KMT2ATSHRCYP1A2CYP2C19
SCHEMBL18040073 0.78 TSHR (0.52) MEN1KMT2ATSHRCYP1A2CYP2C19
SCHEMBL5366626 0.78 ALDH1A1 (0.52) MEN1KMT2ATSHRCYP1A2CYP2C19
SCHEMBL6607473 0.78 NPSR1 (0.52) MEN1KMT2ATSHRCYP1A2CYP2C19
SCHEMBL1465773 0.77 MEN1 (0.54) MEN1KMT2ATSHRCYP1A2CYP2C19
SCHEMBL5644547 0.76 OPRM1 (0.42) GSK3BCA1CA2SIGMAR1ALDH1A1
SCHEMBL1769917 0.76 HSD11B1 (0.51) GSK3BKMT2ALMNAL3MBTL1ALDH1A1
SCHEMBL19207553 0.75 AKR1C1 (0.52) GSK3BMEN1KMT2ALMNANPSR1
SCHEMBL30768288 0.75 ALDH1A1 (0.49) MEN1KMT2ATSHRCYP1A2CYP2C19
SCHEMBL1769341 0.74 LMNA (0.64) MEN1KMT2ATSHRCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115703758-B Compounds used as kinase inhibitors, preparation method and application thereof 中国医学科学院药物研究所 2024-03-26 CN disclosed