SCHEMBL29217023

SCHEMBL29217023

CCc1nc(C(=O)O)cc2c3ccccc3n(Cc3ccc(OC)cc3)c12

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 1/20 0.50
TP53 P04637 2/20 0.48
TSPO P30536 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
CHRM1 P11229 1/20 0.45
FABP4 P15090 1/20 0.45
PLA2G2A P14555 3/20 0.44
CCR2 P41597 2/20 0.44
EDNRB P24530 2/20 0.44
KMT2A Q03164 2/20 0.43
MAPT P10636 1/20 0.43
MEN1 O00255 1/20 0.43
MCL1 Q07820 1/20 0.43
EDNRA P25101 1/20 0.43
TBXA2R P21731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2214735 0.90 CYP19A1 (0.47) P2RX4TP53RXFP1CCR2KMT2A
SCHEMBL29217042 0.89 KDM4E (0.53) P2RX4TP53FABP4CCR2KMT2A
SCHEMBL29217015 0.89 CCR2 (0.48) TP53TSPOCCR2KMT2AMAPT
SCHEMBL29217013 0.88 MEN1 (0.48) TP53TSPOFABP4CCR2KMT2A
SCHEMBL27917551 0.87 KDM4E (0.49) P2RX4TP53TSPOCHRM1KMT2A
SCHEMBL29217030 0.85 FABP4 (0.44) FABP4MAPT
SCHEMBL29217025 0.85 P2RX4 (0.41) P2RX4TP53TSPORXFP1KMT2A
SCHEMBL29217006 0.84 LMNA (0.47) TP53TSPOFABP4EDNRBKMT2A
SCHEMBL27899805 0.83 CNR2 (0.48) TSPO
SCHEMBL2214060 0.82 ALDH1A1 (0.48) RXFP1KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118084903-A Beta-carboline hydrogen sulfide donor derivative and preparation method and application thereof 贵州医科大学 2024-05-28 CN claimed
CN-118084903-A Beta-carboline hydrogen sulfide donor derivative and preparation method and application thereof 贵州医科大学 2024-05-28 CN disclosed