SCHEMBL29234875

SCHEMBL29234875

O=Cn1cc(C(F)(F)F)nc1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 16/20 0.52
PTGS1 P23219 9/20 0.52
HPGD P15428 1/20 0.41
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480252 0.77 PTGS2 (0.54) PTGS2PTGS1HSD17B10
SCHEMBL27855491 0.77 OGG1 (0.40) HPGDKDM4EHSD17B10LMNAPOLB
SCHEMBL13437655 0.76 PTGS2 (0.72) PTGS2PTGS1
SCHEMBL11622203 0.75 PTGS2 (0.51) PTGS2PTGS1KDM4EHSD17B10
SCHEMBL7469586 0.72 PTGS2 (0.46) PTGS2PTGS1HPGDKDM4ELMNA
Sulfamide SCHEMBL4639731 0.72 PTGS2 (0.82) PTGS2PTGS1
SCHEMBL11623751 0.71 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL14278512 0.70 PTGS2 (0.67) PTGS2PTGS1
SCHEMBL215075 0.69 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL215038 0.69 PTGS2 (1.00) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115557904-B Synthetic method suitable for large-scale production of 5, 7-bis (trifluoromethyl) quinazoline-2, 4-dione 天津药明康德新药开发有限公司 2024-03-19 CN claimed
CN-115557904-B Synthetic method suitable for large-scale production of 5, 7-bis (trifluoromethyl) quinazoline-2, 4-dione 天津药明康德新药开发有限公司 2024-03-19 CN disclosed