SCHEMBL2923724

SCHEMBL2923724

COc1ncnc2sc(NC(=O)ON3CCN(CCOc4cccc(C(F)(F)F)c4)CC3)nc12

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
ADORA2A P29274 1/20 0.40
DRD2 P14416 5/20 0.40
LTA4H P09960 1/20 0.40
HTR1A P08908 1/20 0.39
HTR7 P34969 1/20 0.39
EPHX2 P34913 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
SCD O00767 1/20 0.39
HTR2A P28223 1/20 0.38
DRD3 P35462 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1760945 0.89 LMNA (0.47) KDM4EALDH1A1LMNAGAAHTT
SCHEMBL2927982 0.87 ADORA2B (0.47) KDM4EALDH1A1GAAKMT2AADORA2A
SCHEMBL3041508 0.84 PHGDH (0.47) ALDH1A1LMNAGAAHTTKMT2A
SCHEMBL2932276 0.83 CYP2D6 (0.41) ALDH1A1ADORA2A
SCHEMBL3039094 0.82 TACR1 (0.36) ADORA2ASCD
SCHEMBL2925605 0.82 FAAH (0.40) ALDH1A1LMNAGAAKMT2ADRD2
SCHEMBL2930871 0.82 ADORA2A (0.49) HTTADORA2ADRD2
SCHEMBL2931360 0.81 GPR6 (0.47) ADORA2ADRD2
SCHEMBL2932713 0.81 ADORA2A (0.49) KDM4EALDH1A1LMNAGAAHTT
SCHEMBL2931382 0.81 ADORA2A (0.41) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed