SCHEMBL29239267

SCHEMBL29239267

CN1C(=O)C2CNCCN2c2ccc(N3C=CC=NC3)cc21

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 17/20 0.36
HTR2A P28223 7/20 0.33
CYP2D6 P10635 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTR2B P41595 7/20 0.32
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11456017 0.72 HTR2C (0.49) HTR2CHTR2ACYP2D6ALDH1A1CYP1A2
SCHEMBL26915074 0.71 HTR2C (0.47) HTR2CHTR2ACYP3A4HTR2B
SCHEMBL26915066 0.71 HTR2C (0.47) HTR2CHTR2ACYP3A4HTR2B
SCHEMBL30729654 0.71 HTR2C (0.47) HTR2CHTR2ACYP3A4HTR2B
Hydrochloric Acid SCHEMBL6421986 0.71 HTR2C (0.49) HTR2CHTR2ACYP2D6ALDH1A1CYP1A2
SCHEMBL27039628 0.69 HTR3A (0.47) HTR2B
SCHEMBL29114220 0.68 THRB (0.40) HTR2CHTR2ACYP2D6ALDH1A1CYP1A2
SCHEMBL29239264 0.67 PRKCQ (0.43) HTR2C
SCHEMBL29239265 0.67 PRKCQ (0.43) HTR2C
SCHEMBL27039521 0.64 ADRB2 (0.51) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118005655-A Condensed ring compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2024-05-10 CN disclosed