SCHEMBL2927062

SCHEMBL2927062

COc1ccc(S(=O)(=O)N2[C@H]3CN(C(=O)O)CC[C@H]3C[C@]2(Cc2ccccc2)C(=O)NO)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 14/20 0.51
MMP2 P08253 2/20 0.51
MMP12 P39900 1/20 0.51
MMP1 P03956 14/20 0.46
MMP3 P08254 8/20 0.46
MMP7 P09237 7/20 0.46
MMP8 P22894 1/20 0.46
MMP13 P45452 11/20 0.46
ADAM17 P78536 3/20 0.45
PKM P14618 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GRIN2B Q13224 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2927853 0.90 MMP9 (0.47) MMP9MMP2MMP12MMP1MMP3
SCHEMBL1658411 0.87 MMP9 (0.45) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2928560 0.77 MMP9 (0.52) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927569 0.77 MMP9 (0.50) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2929201 0.76 MMP9 (0.46) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2928574 0.73 MMP9 (0.49) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927547 0.70 MMP9 (0.75) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2927653 0.70 MMP9 (0.68) MMP9MMP2MMP12MMP1MMP3
SCHEMBL2930771 0.69 ALDH1A1 (0.43) PKM
SCHEMBL5546935 0.68 MMP9 (0.61) MMP9MMP2MMP12MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768979-B1 OCTAHYDROPYRROLO[2, 3, C]PYRIDINE DERIVATIVES AND PHARMACEUTICAL USE THEREOF MERCK SERONO SA (CH) 2010-09-29 EP claimed