SCHEMBL2927231

SCHEMBL2927231

CCOC(=O)[C@@](C)(NC(=O)OC(C)(C)C)c1ccccc1Br

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 2/20 0.41
RECQL P46063 1/20 0.41
MMP8 P22894 1/20 0.41
PTPRB P23467 1/20 0.41
AAK1 Q2M2I8 3/20 0.40
PIN1 Q13526 1/20 0.40
AKT1 P31749 2/20 0.39
SYK P43405 1/20 0.38
CTSS P25774 1/20 0.38
CTSK P43235 1/20 0.38
F2R P25116 1/20 0.38
MAPT P10636 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3004859 0.82 MEN1 (0.47) KMT2AMEN1NPC1HTTRAB9A
SCHEMBL2929698 0.80 KMT2A (0.38) KMT2AMEN1HTTALDH1A1RECQL
SCHEMBL24045987 0.78 PIN1 (0.47) KMT2AMEN1ALDH1A1RECQLMMP8
SCHEMBL4542373 0.77 PTPRB (0.39) KMT2AMEN1NPC1HTTRAB9A
SCHEMBL2923484 0.76 PIN1 (0.41) KMT2AMEN1NPC1HTTRAB9A
SCHEMBL2490507 0.74 ABCB11 (0.49) KMT2AALDH1A1RECQLPTPRBMAPT
SCHEMBL7233451 0.74 PTPRB (0.45) NPC1RAB9AALDH1A1RECQLMMP8
SCHEMBL2925457 0.74 PTPRB (0.42) KMT2AMEN1ALDH1A1RECQLMMP8
SCHEMBL31619484 0.74 PIN1 (0.46) KMT2AMEN1HTTALDH1A1RECQL
SCHEMBL1509032 0.73 KMT2A (0.44) KMT2AMEN1NPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225253-A1 PHOSPHONIC ACID DERIVATES AND THEIR USE AS P2Y12 RECEPTOR ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2010-09-08 EP disclosed
WO-2009069100-A1 PHOSPHONIC ACID DERIVATES AND THEIR USE AS P2Y12 RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2009-06-04 WO disclosed