SCHEMBL29282154

SCHEMBL29282154

NC1=NCc2c(B(O)O)cccc21

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
NOS2 P35228 2/20 0.34
NOS3 P29474 2/20 0.34
HTR5A P47898 2/20 0.33
F9 P00740 1/20 0.30
HTR1A P08908 1/20 0.30
HTR1D P28221 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR7 P34969 1/20 0.30
HTR3A P46098 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8736593 0.72 HTR5A (0.50) TSHRNOS2NOS3HTR5A
SCHEMBL10033961 0.63 NPC1 (0.50) HTR2CHTR7
SCHEMBL29955280 0.63 KCNJ1 (0.49)
SCHEMBL17132729 0.62 ENPP2 (0.41)
SCHEMBL31703623 0.62 TSHR (0.95) TSHRNOS2NOS3HTR5A
SCHEMBL1194687 0.62 TSHR (0.95) TSHRNOS2NOS3HTR5A
SCHEMBL8487986 0.62 NOS2 (0.52) TSHRNOS2NOS3HTR5A
SCHEMBL27632016 0.62 CES1 (0.41) HTR1AHTR1DHTR2AHTR7HTR3A
SCHEMBL910658 0.61 ENPP2 (0.50)
SCHEMBL2144193 0.61 CLK4 (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117986241-A Biphenyl derivative, pharmaceutical composition and application thereof 武汉睿健医药科技有限公司 2024-05-07 CN disclosed