SCHEMBL2928449

SCHEMBL2928449

COc1ncnc2sc(NC(=O)ON3CCN(Cc4cccc(OC(F)F)c4)CC3)nc12

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 4/20 0.46
FAAH O00519 4/20 0.39
ACHE P22303 1/20 0.38
ALDH1A1 P00352 3/20 0.38
LPAR2 Q9HBW0 1/20 0.38
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
PHGDH O43175 1/20 0.37
PDE2A O00408 1/20 0.37
GAA P10253 2/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2930504 0.93 FAAH (0.45) GPR6FAAHALDH1A1KDM4EMEN1
SCHEMBL2931360 0.92 GPR6 (0.47) GPR6FAAHACHE
SCHEMBL2925605 0.89 FAAH (0.40) GPR6FAAHACHEALDH1A1LPAR2
SCHEMBL1760954 0.89 FAAH (0.49) GPR6FAAHALDH1A1KDM4EMEN1
SCHEMBL2931169 0.88 OGA (0.38) GPR6FAAHACHELPAR2MEN1
SCHEMBL3049811 0.87 MEN1 (0.42) FAAHACHEALDH1A1LPAR2MEN1
SCHEMBL2929411 0.87 ADORA2A (0.41) ACHEALDH1A1KDM4EMEN1HTT
SCHEMBL2927982 0.87 ADORA2B (0.47) FAAHALDH1A1KDM4EMEN1KMT2A
SCHEMBL2930506 0.86 GPR6 (0.38) GPR6ACHEALDH1A1MEN1KMT2A
SCHEMBL2931204 0.85 GPR6 (0.47) GPR6FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2027132-B1 THIAZOLO-PYRAMIDINE / PYRIDINE UREA DERIVATIVES AS ADENOSINE A2B RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2010-09-15 EP claimed