SCHEMBL2928469

SCHEMBL2928469

Nc1nccc(Oc2ccc(NC(=O)O)cc2F)c1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MET P08581 20/20 0.49
KDR P35968 3/20 0.49
RET P07949 1/20 0.49
KIT P10721 1/20 0.49
PDGFRA P16234 1/20 0.49
FLT3 P36888 1/20 0.49
CYP3A4 P08684 2/20 0.45
AXL P30530 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2928468 1.00 MET (0.49) METKDRRETKITPDGFRA
SCHEMBL13610912 0.89 MET (0.47) METKDRRETKITPDGFRA
SCHEMBL4464910 0.88 SMN1; SMN2 (0.42) METKDRRETKITPDGFRA
SCHEMBL4464904 0.88 SMN1; SMN2 (0.42) METKDRRETKITPDGFRA
SCHEMBL3762191 0.86 MET (0.45) METKDRRETKITPDGFRA
SCHEMBL29988424 0.86 MET (0.45) METKDRRETKITPDGFRA
SCHEMBL3842300 0.86 LMNA (0.48) METKDRRETKITPDGFRA
SCHEMBL3842301 0.86 LMNA (0.48) METKDRRETKITPDGFRA
SCHEMBL2934893 0.84 MET (0.54) METKDRRETKITPDGFRA
SCHEMBL18256938 0.83 MET (0.74) METKDRRETKITPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229391-A1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE Cancer Research Technology Limited (GB) 2010-09-22 EP disclosed
WO-2009077766-A1 PYRIDO[2,3-B]PYRAZINE-8-SUBSTITUTED COMPOUNDS AND THEIR USE CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2009-06-25 WO disclosed