SCHEMBL29295115

SCHEMBL29295115

O=c1[nH]c(N2CCOCC2)nc2nn(-c3c(F)cc(C4CC4)cc3C(F)(F)F)cc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.40
PDE3B Q13370 4/20 0.37
PDE3A Q14432 4/20 0.37
KMT2A Q03164 2/20 0.34
IRAK4 Q9NWZ3 5/20 0.34
PIK3CA P42336 2/20 0.33
PIK3CD O00329 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
SCD O00767 1/20 0.33
TSHR P16473 2/20 0.32
PIK3R1 P27986 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
MEN1 O00255 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MGLL Q99685 1/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29294901 0.90 NLRP3 (0.45) NLRP3PDE3BPDE3AKMT2AIRAK4
SCHEMBL29294075 0.88 NLRP3 (0.49) NLRP3PDE3BPDE3AKMT2AIRAK4
SCHEMBL29295113 0.86 NLRP3 (0.50) NLRP3PDE3BPDE3AKMT2APIK3CA
SCHEMBL29294905 0.85 PDE3B (0.39) NLRP3PDE3BPDE3AKMT2AIRAK4
SCHEMBL31367978 0.83 PDE3B (0.38) PDE3BPDE3AKMT2AIRAK4PIK3CA
SCHEMBL29294065 0.82 NLRP3 (0.53) NLRP3KMT2AIRAK4TSHRALDH1A1
SCHEMBL29295243 0.79 NLRP3 (0.50) NLRP3KMT2AIRAK4TSHRALDH1A1
SCHEMBL29294923 0.79 NLRP3 (0.42) NLRP3PDE3BPDE3AKMT2ATSHR
SCHEMBL29295109 0.79 NLRP3 (0.52) NLRP3KMT2AIRAK4TSHRALDH1A1
SCHEMBL29294899 0.79 NLRP3 (0.58) NLRP3PDE3BPDE3AKMT2APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4397663-A1 6-AMINOPYRAZOLOPYRIMIDINE COMPOUND AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2024-07-10 EP disclosed