SCHEMBL2931080

SCHEMBL2931080

COc1ccc(-c2ccccc2C(=O)N2C[C@H]3C[C@H]3[C@H]2CN)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 9/20 0.42
HCRTR2 O43614 7/20 0.42
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40
TUBA4A P68366 1/20 0.40
TUBB4B P68371 1/20 0.40
TUBB3 Q13509 1/20 0.40
TUBB2A Q13885 1/20 0.40
TUBB8 Q3ZCM7 1/20 0.40
TUBA3E Q6PEY2 1/20 0.40
TUBA1A Q71U36 1/20 0.40
TUBA1C Q9BQE3 1/20 0.40
TUBB6 Q9BUF5 1/20 0.40
TUBB2B Q9BVA1 1/20 0.40
TUBB1 Q9H4B7 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
MMP1 P03956 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2929170 0.89 KDM4E (0.43) HCRTR1HCRTR2GAACDK4CCND1
SCHEMBL2931897 0.88 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL3417003 0.88 HCRTR1 (0.45) HCRTR1HCRTR2
SCHEMBL3415643 0.88 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2930541 0.88 HCRTR1 (0.46) HCRTR1HCRTR2
SCHEMBL2925288 0.87 HCRTR1 (0.46) HCRTR1HCRTR2CDK4CCND1MLNR
SCHEMBL3415834 0.87 HCRTR1 (0.46) HCRTR1HCRTR2CDK4CCND1MLNR
SCHEMBL2924532 0.86 SLC6A4 (0.40) HCRTR1HCRTR2MLNRCYP3A4
SCHEMBL2931078 0.84 FPR2 (0.41) HCRTR1HCRTR2TUBB4ATUBBTUBA3C
SCHEMBL2446753 0.83 HCRTR1 (0.42) HCRTR1HCRTR2GAACDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP claimed
EP-2079690-B1 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2010-09-15 EP disclosed