SCHEMBL29313615

SCHEMBL29313615

CNc1ncc(C#N)c(NCc2cccnn2)n1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 4/20 0.47
PTK2 Q05397 1/20 0.43
PTK2B Q14289 1/20 0.43
SYK P43405 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
HSD17B10 Q99714 1/20 0.36
AURKA O14965 1/20 0.36
SIRT5 Q9NXA8 1/20 0.36
PRKCQ Q04759 7/20 0.36
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
KMT2A Q03164 1/20 0.35
LRRK2 Q5S007 2/20 0.34
PGK1 P00558 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29313537 0.85 PTK2 (0.56) PTK2PTK2BSYKMEN1ALDH1A1
SCHEMBL29313552 0.80 PTK2 (0.43) VNN1PTK2PTK2BSYKCYP1A2
SCHEMBL29313606 0.80 PTK2 (0.40) PTK2PTK2BSYKAURKASIRT5
SCHEMBL29313621 0.80 PTK2 (0.41) PTK2PTK2BSYKCYP1A2CYP3A4
SCHEMBL29313542 0.80 ALDH1A1 (0.54) VNN1CYP1A2CYP3A4TDP1HSD17B10
SCHEMBL29315070 0.75 MAP3K8 (0.45) PTK2PTK2BSYKAURKASIRT5
SCHEMBL29315097 0.73 MAP3K8 (0.43) PTK2PTK2BSYKAURKASIRT5
SCHEMBL29313773 0.71 CCNA2 (0.46) SYKAURKASIRT5PRKCQALDH1A1
SCHEMBL18419810 0.69 APP (0.48) PTK2PTK2BCYP1A2TDP1HSD17B10
SCHEMBL29315063 0.69 LRRK2 (0.35) SYKAURKASIRT5PRKCQLRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed