SCHEMBL29313852

SCHEMBL29313852

CN(C(=O)Oc1c(-n2cc[nH]c2=S)cc(C(F)(F)F)cc1C(F)(F)F)c1ccc(F)cc1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
POLQ O75417 5/20 0.41
LIPE Q05469 5/20 0.32
ALDH1A1 P00352 3/20 0.32
SCN8A Q9UQD0 2/20 0.32
SCN10A Q9Y5Y9 2/20 0.32
TACR1 P25103 1/20 0.32
KMT2A Q03164 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31009145 0.90 POLQ (0.44) POLQLIPESCN8ASCN10AKMT2A
SCHEMBL29314474 0.90 POLQ (0.44) POLQLIPESCN8ASCN10AKMT2A
SCHEMBL29314303 0.88 POLQ (0.33) POLQALDH1A1SCN8ASCN10ATACR1
SCHEMBL31009165 0.84 POLQ (0.46) POLQSCN8ASCN10A
SCHEMBL29313853 0.83 ALDH1A1 (0.31) ALDH1A1
SCHEMBL29313854 0.83 POLB (0.31)
SCHEMBL29313855 0.83 POLQ (0.37) POLQ
SCHEMBL29313860 0.82 POLQ (0.34) POLQ
SCHEMBL29313609 0.78 POLQ (0.40) POLQLIPE
SCHEMBL29314384 0.78 POLQ (0.52) POLQLIPEALDH1A1TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed