SCHEMBL29314407

SCHEMBL29314407

CNc1ncc(C#N)c(N(C)CC(C)(C)O)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.36
KDR P35968 3/20 0.36
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
PLK1 P53350 2/20 0.32
LRRK2 Q5S007 5/20 0.32
AURKA O14965 1/20 0.32
CCNT1 O60563 2/20 0.31
CDK2 P24941 2/20 0.31
CDK9 P50750 2/20 0.31
CCNA2 P20248 1/20 0.31
CCNA1 P78396 1/20 0.31
AR P10275 1/20 0.31
NUDT1 P36639 2/20 0.31
CDK4 P11802 1/20 0.31
CCNB1 P14635 1/20 0.31
CCND1 P24385 1/20 0.31
CCNE1 P24864 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2540599 0.68 MAPK14 (0.57) MAPK13MAPK12MAPK11MAPK14LRRK2
SCHEMBL13523666 0.67 KDM4E (0.41) CDK1KDRLRRK2AURKACCNT1
SCHEMBL4769052 0.66 CSNK1A1 (0.44) ARNUDT1
SCHEMBL29314042 0.66 NUDT1 (0.45) CDK1KDRLRRK2AURKANUDT1
SCHEMBL25598891 0.66 CSNK1A1 (0.42) CDK1KDRLRRK2AURKACCNT1
SCHEMBL29313773 0.64 CCNA2 (0.46) CDK1KDRLRRK2AURKACDK2
SCHEMBL25597187 0.63 IDH1 (0.45) CDK1KDRLRRK2
SCHEMBL29313462 0.62 LRRK2 (0.39) LRRK2AURKACHEK1
SCHEMBL13587064 0.62 AURKA (0.37) CDK1KDRLRRK2AURKACCNT1
SCHEMBL29313821 0.62 PLK1 (0.39) KDRPLK1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed