SCHEMBL29314691

SCHEMBL29314691

CNc1ncc(C#N)c(-c2cccc(F)c2)n1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 8/20 0.63
ADORA2B P29275 3/20 0.63
KDR P35968 7/20 0.51
CDK1 P06493 4/20 0.49
CHUK O15111 1/20 0.46
ADORA2A P29274 4/20 0.45
HSP90AB1 P08238 1/20 0.44
MERTK Q12866 1/20 0.44
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 1/20 0.43
RAB9A P51151 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314862 0.78 ADORA1 (0.64) ADORA1ADORA2BKDRCDK1ADORA2A
SCHEMBL24478143 0.77 CDK1 (0.62) KDRCDK1RAB9A
SCHEMBL5451373 0.75 ADORA1 (0.53) ADORA1ADORA2BADORA2AMERTK
SCHEMBL29315373 0.75 KDR (0.48) ADORA1KDRCDK1ADORA2AMERTK
SCHEMBL29314783 0.74 KDR (0.47) ADORA1ADORA2BKDRCDK1ADORA2A
SCHEMBL5452581 0.74 ADORA1 (0.48) ADORA1ADORA2BADORA2AMERTK
SCHEMBL4221233 0.74 MERTK (0.62) ADORA1ADORA2BMERTK
SCHEMBL15832010 0.73 ADORA1 (0.49) ADORA1ADORA2BCHUKADORA2AALDH1A1
SCHEMBL6033274 0.72 KDR (0.62) KDRCDK1
SCHEMBL29314732 0.71 KDR (0.61) ADORA1KDRCDK1CHUKADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed