SCHEMBL29314788

SCHEMBL29314788

CC1(C)OB(c2ccc(C(F)(F)F)cc2C(F)(F)F)OC1(C)C

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.39
LIPE Q05469 6/20 0.37
LPL P06858 4/20 0.34
LIPG Q9Y5X9 4/20 0.34
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
F2 P00734 1/20 0.31
F11 P03951 1/20 0.31
PRSS1 P07477 1/20 0.31
PRSS2 P07478 1/20 0.31
PRSS3 P35030 1/20 0.31
POLQ O75417 2/20 0.31
AR P10275 1/20 0.31
PDE2A O00408 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30847591 1.00 CES2 (0.39) CES2LIPELPLLIPGPDE4A
SCHEMBL17903423 0.87 LIPE (0.35) CES2LIPE
SCHEMBL31207708 0.87 LIPE (0.35) CES2LIPE
SCHEMBL837370 0.85 LIPE (0.39) LIPELPLLIPGPDE4APDE4B
SCHEMBL19031772 0.83 LPL (0.45) LPLLIPGF2F11PRSS1
SCHEMBL29909454 0.83 PDE2A (0.39) LIPELPLLIPGPDE4APDE4B
SCHEMBL20536870 0.83 LPL (0.45) LPLLIPGF2F11PRSS1
SCHEMBL4108381 0.83 PDE2A (0.39) LIPELPLLIPGPDE4APDE4B
SCHEMBL22606823 0.82 LPL (0.36) LIPELPLLIPGF2F11
SCHEMBL24596359 0.82 ALDH1A1 (0.39) LIPELPLLIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed