SCHEMBL29314803

SCHEMBL29314803

CNc1ncc(C#N)c(-c2cnn(CC(N)=O)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 8/20 0.46
CCNT1 O60563 4/20 0.46
CDK4 P11802 4/20 0.46
CCNB1 P14635 4/20 0.46
CCND1 P24385 4/20 0.46
CCNE1 P24864 4/20 0.46
CDK2 P24941 4/20 0.46
CCND3 P30281 4/20 0.46
CDK7 P50613 4/20 0.46
CDK9 P50750 4/20 0.46
CCNH P51946 4/20 0.46
MNAT1 P51948 4/20 0.46
CDK6 Q00534 4/20 0.46
KDM5A P29375 1/20 0.38
KDM5C P41229 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
EP300 Q09472 2/20 0.38
JAK2 O60674 5/20 0.37
JAK1 P23458 5/20 0.37
JAK3 P52333 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29314874 0.80 CDK1 (0.56) CDK1CCNT1CDK4CCNB1CCND1
SCHEMBL29315373 0.69 KDR (0.48) CDK1CCNT1CDK2CDK9KDR
SCHEMBL30291335 0.68 CDK1 (0.59) CDK1CCNT1CDK4CCNB1CCND1
SCHEMBL29314732 0.68 KDR (0.61) CDK1CCNT1CCNB1CDK2CDK7
SCHEMBL31121901 0.68 CDK1 (0.67) CDK1CCNT1CDK4CCNB1CCND1
SCHEMBL21596384 0.66 KDM5A (0.38) CDK1CCNT1CDK4CCNB1CCND1
SCHEMBL21600836 0.65 KDM5A (0.37) CDK1CCNT1CDK4CCNB1CCND1
SCHEMBL29314862 0.65 ADORA1 (0.64) CDK1KDR
SCHEMBL30291202 0.64 CDK1 (0.58) CDK1CCNT1CDK4CCNB1CCND1
SCHEMBL29314691 0.63 ADORA1 (0.63) CDK1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed