SCHEMBL29315437

SCHEMBL29315437

Cc1cc(-c2nc(N)ncc2C#N)[nH]n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.49
ADORA2A P29274 1/20 0.49
CSNK1A1 P48729 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
CDK4 P11802 1/20 0.33
CCND3 P30281 1/20 0.33
P2RX3 P56373 1/20 0.33
P2RX2 Q9UBL9 1/20 0.33
LRRK2 Q5S007 1/20 0.32
CDK1 P06493 3/20 0.32
KDR P35968 3/20 0.32
PLK4 O00444 1/20 0.32
CHEK1 O14757 1/20 0.32
AURKA O14965 1/20 0.32
CHUK O15111 1/20 0.32
ROCK2 O75116 1/20 0.32
CHEK2 O96017 1/20 0.32
INSR P06213 1/20 0.32
CSF1R P07333 1/20 0.32
PIM1 P11309 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4464801 0.74 DHFR (0.42) ADORA1FGFR1
SCHEMBL18356737 0.70 ADORA1 (0.71) ADORA1ADORA2ACDK1KDRCHUK
SCHEMBL1579901 0.69 ADORA2A (0.51) ADORA1ADORA2ACSNK1A1CLK4CDK4
SCHEMBL3361914 0.68 ADORA2A (0.51) ADORA1ADORA2A
SCHEMBL15722386 0.66 ADORA2A (0.43) ADORA1ADORA2ALRRK2CHUKCDK2
SCHEMBL6034022 0.66 ADORA1 (1.00) ADORA1ADORA2ACDK1KDRCHUK
SCHEMBL23019354 0.66 TRPA1 (0.56) ADORA1ADORA2ACLK4KDRROCK2
SCHEMBL29313431 0.66 ADORA2A (0.60) ADORA1ADORA2ACSNK1A1CLK4CDK1
SCHEMBL263835 0.65 CSNK1A1 (0.64) ADORA1ADORA2ACSNK1A1CLK4P2RX3
SCHEMBL6446312 0.65 ADORA2A (0.57) ADORA1ADORA2AP2RX3P2RX2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3782986-B1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICALS CO (JP) 2024-07-10 EP disclosed