SCHEMBL29315902

SCHEMBL29315902

O=C(O)Cc1c(Br)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 8/20 0.44
RXRG P48443 8/20 0.44
RXRB P28702 7/20 0.44
GPR17 Q13304 1/20 0.42
AGBL2 Q5U5Z8 1/20 0.40
CES2 O00748 1/20 0.39
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
LMNA P02545 1/20 0.37
NOTUM Q6P988 1/20 0.37
AKR1B1 P15121 1/20 0.37
EGLN1 Q9GZT9 1/20 0.36
NR3C1 P04150 1/20 0.36
THRB P10828 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315906 0.81 NOTUM (0.47) RXRARXRGRXRBCES2LMNA
SCHEMBL15524368 0.75 AKR1B1 (0.43) RXRARXRGRXRBLMNAAKR1B1
SCHEMBL6864341 0.74 CES2 (0.46) RXRARXRGRXRBGPR17CES2
SCHEMBL29009799 0.73 RXRA (0.50) RXRARXRGRXRBGPR17AGBL2
SCHEMBL2184606 0.72 RXRA (0.54) RXRARXRGRXRBAGBL2PSEN1
SCHEMBL2525416 0.72 AKR1B1 (0.52) RXRARXRGRXRBAGBL2CES2
SCHEMBL15524659 0.71 RXRA (0.50) RXRARXRGRXRBAGBL2CES2
SCHEMBL509209 0.70 RXRA (0.49) RXRARXRGRXRBAGBL2CES2
SCHEMBL6096516 0.70 RXRA (0.52) RXRARXRGRXRBGPR17AGBL2
SCHEMBL7584232 0.69 RXRA (0.39) RXRARXRGRXRBGPR17AGBL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed