SCHEMBL29315906

SCHEMBL29315906

COC(=O)Cc1c(Br)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.47
AKR1C3 P42330 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 3/20 0.36
XBP1 P17861 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HSP90AB1 P08238 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
GPR35 Q9HC97 2/20 0.35
ACP1 P24666 1/20 0.35
CES2 O00748 1/20 0.35
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
KDM4E B2RXH2 2/20 0.34
CACNA1H O95180 1/20 0.34
CACNA1B Q00975 1/20 0.34
CACNA1C Q13936 1/20 0.34
SOS1 Q07889 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29315902 0.81 RXRA (0.44) NOTUMLMNAMAPTXBP1NPSR1
SCHEMBL15524632 0.78 NOTUM (0.43) NOTUMLMNAMAPTMEN1KMT2A
SCHEMBL23531156 0.76 NOTUM (0.56) NOTUMLMNAHSP90AB1MEN1KMT2A
SCHEMBL15524663 0.75 CFTR (0.43) NOTUMAKR1C3LMNAMAPTMEN1
SCHEMBL29315909 0.73 ROCK2 (0.46)
SCHEMBL29823794 0.73 NOTUM (0.36) NOTUMCACNA1H
SCHEMBL1296063 0.73 HSP90AB1 (0.56) NOTUMLMNAMAPTHSP90AB1CES2
SCHEMBL15524132 0.72 PPARG (0.44) NOTUMAKR1C3LMNAMAPTXBP1
SCHEMBL14661309 0.72 P2RX7 (0.45) LMNAMAPTHSP90AB1MEN1KMT2A
SCHEMBL18524127 0.72 NOTUM (0.57) NOTUMLMNAMAPTHSP90AB1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed