SCHEMBL7584232

SCHEMBL7584232

C=CCCc1c(CC(=O)O)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RXRA P19793 9/20 0.39
RXRG P48443 9/20 0.39
RXRB P28702 8/20 0.39
GPR17 Q13304 1/20 0.39
AGBL2 Q5U5Z8 1/20 0.34
POLQ O75417 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
CES2 O00748 1/20 0.33
EGLN1 Q9GZT9 1/20 0.32
LMNA P02545 1/20 0.32
PTGS2 P35354 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6096516 0.72 RXRA (0.52) RXRARXRGRXRBGPR17AGBL2
SCHEMBL8462688 0.70 RXRA (0.43) RXRARXRGRXRBGPR17AGBL2
SCHEMBL8464813 0.70 RXRA (0.43) RXRARXRGRXRBGPR17AGBL2
SCHEMBL29315902 0.69 RXRA (0.44) RXRARXRGRXRBGPR17AGBL2
SCHEMBL5574328 0.68 CES2 (0.53) RXRARXRGRXRBAGBL2POLQ
SCHEMBL30716953 0.68 POLQ (0.61) RXRARXRGRXRBPOLQPTGDR2
SCHEMBL3741058 0.68 POLQ (0.61) RXRARXRGRXRBPOLQPTGDR2
SCHEMBL30428330 0.67 RXRA (0.50) RXRARXRGRXRBAGBL2PTGDR2
SCHEMBL6864341 0.67 CES2 (0.46) RXRARXRGRXRBGPR17POLQ
SCHEMBL509209 0.66 RXRA (0.49) RXRARXRGRXRBAGBL2PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002102372-A1 GEM-DISUBSTITUTED CYCLOHEXANE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2002-12-27 WO disclosed