SCHEMBL29316723

SCHEMBL29316723

CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
CES2 O00748 3/20 0.39
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
NOTUM Q6P988 1/20 0.38
PTPN5 P54829 1/20 0.37
HSPA5 P11021 1/20 0.37
POLQ O75417 3/20 0.36
GPR35 Q9HC97 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
P2RX1 P51575 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9861458 0.88 GABRA1 (0.50) ESR1ESR2CES2GABRA1GABRB2
SCHEMBL30055403 0.82 SIRT2 (0.41) CES2POLQ
SCHEMBL9862041 0.81 HSPA5 (0.58) GABRA1GABRB2PTPN5HSPA5SIGMAR1
SCHEMBL18244651 0.81 CACNA1H (0.36) CES2
SCHEMBL13888158 0.79 GABRB3 (0.41) ESR1ESR2GABRA1GABRB2GPR35
SCHEMBL13888162 0.79 GABRA1 (0.38) GABRA1GABRB2PTPN5HSPA5POLQ
SCHEMBL391593 0.79 CES2 (0.45) CES2NOTUMGPR35
SCHEMBL6909178 0.77 CES2 (0.40) CES2NOTUMPOLQGPR35SIGMAR1
SCHEMBL424607 0.77 POLQ (0.40) CES2NOTUMPOLQGPR35SIGMAR1
SCHEMBL16772949 0.75 CYP1A2 (0.43) ESR1ESR2CES2GABRA1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed