SCHEMBL6909178

SCHEMBL6909178

CCc1cc(C(F)(F)F)cc(C(F)(F)F)c1C(C)=O

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.40
NOTUM Q6P988 1/20 0.38
POLQ O75417 3/20 0.37
GPR35 Q9HC97 1/20 0.36
SIGMAR1 Q99720 3/20 0.36
RXRA P19793 2/20 0.35
RXRB P28702 2/20 0.35
RXRG P48443 2/20 0.35
MAOB P27338 1/20 0.35
CACNA1H O95180 1/20 0.34
MAPT P10636 1/20 0.34
KIF11 P52732 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424607 0.86 POLQ (0.40) CES2NOTUMPOLQGPR35SIGMAR1
SCHEMBL30628783 0.85 CES2 (0.47) CES2NOTUMPOLQGPR35RXRA
SCHEMBL3024423 0.85 CES2 (0.39) CES2NOTUMPOLQGPR35SIGMAR1
SCHEMBL6910600 0.79 KIF11 (0.42) CES2NOTUMPOLQRXRARXRB
SCHEMBL2308100 0.78 CES2 (0.42) CES2NOTUMGPR35RXRARXRB
SCHEMBL29316723 0.77 ESR1 (0.39) CES2NOTUMPOLQGPR35SIGMAR1
SCHEMBL2313613 0.74 KDM4E (0.45) CES2NOTUMGPR35RXRARXRB
SCHEMBL18378522 0.73 CES2 (0.41) CES2NOTUMGPR35CACNA1HMAPT
SCHEMBL12439666 0.72 RXRA (0.40) CES2GPR35SIGMAR1RXRARXRB
SCHEMBL6908816 0.72 IDO1 (0.38) CES2CACNA1H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011023667-A1 CARBOCYCLIC GLYT1 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2011-03-03 WO disclosed