SCHEMBL29316732

SCHEMBL29316732

Oc1c(-n2cncn2)cc(C(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
KDM4E B2RXH2 2/20 0.40
GAA P10253 1/20 0.40
BLM P54132 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
CYP3A4 P08684 1/20 0.35
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NTRK1 P04629 1/20 0.33
GRM7 Q14831 2/20 0.33
MAPK10 P53779 1/20 0.32
CNR1 P21554 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25408423 0.72 CNR1 (0.42) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL21849203 0.72 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL31053865 0.71 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL25024965 0.71 ALDH1A1 (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL391593 0.70 CES2 (0.45) ALDH1A1SMN1; SMN2
SCHEMBL17093084 0.70 ALDH1A1 (0.39) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL8183530 0.70 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL9831326 0.69 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL12391448 0.69 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19MAPT
SCHEMBL30847664 0.68 MAPT (0.39) ALDH1A1MAPTHPGDKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed