SCHEMBL29316983

SCHEMBL29316983

O=c1[nH]c2cc(C(F)(F)F)cc(C(F)(F)F)c2o1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1H O95180 10/20 0.39
CACNA1C Q13936 3/20 0.39
CACNA1B Q00975 3/20 0.39
GPR17 Q13304 1/20 0.37
CACNA1G O43497 3/20 0.35
EGLN1 Q9GZT9 3/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
MAPT P10636 1/20 0.34
NOTUM Q6P988 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8873678 0.83 CACNA1H (0.37) CACNA1HCACNA1CCACNA1BGPR17CACNA1G
SCHEMBL13090751 0.81 NOS1 (0.45) NOTUM
SCHEMBL1331615 0.70 NOS1 (0.56) MAPTNOTUM
SCHEMBL8569885 0.69 KMO (0.41) GPR17EGLN1MAOAMAOBNOTUM
SCHEMBL2418890 0.68 CACNA1H (0.41) CACNA1HCACNA1CCACNA1BGPR17CACNA1G
SCHEMBL7779818 0.68 GRIN1 (0.46) CACNA1HCACNA1CCACNA1BGPR17CACNA1G
SCHEMBL29442143 0.68 MAPT (0.54) MAOAMAOBMAPT
SCHEMBL10619033 0.68 MAPT (0.54) MAOAMAOBMAPT
SCHEMBL8873358 0.67 GPR17 (0.47) CACNA1HCACNA1CCACNA1BGPR17CACNA1G
SCHEMBL17260679 0.67 NOS1 (0.56) MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024147972-A2 DNA POLYMERASE THETA INHIBITORS CONTAINING NON-SATURATED 5-MEMBERED HETEROCYCLIC RINGS AND USE THEREOF THOMAS JEFFERSON UNIVERSITY (US) 2024-07-11 WO disclosed