SCHEMBL2933385

SCHEMBL2933385

Brc1cncc(OCCN2CCCCCC2)c1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.56
CHRNA4 P43681 2/20 0.56
KDM4E B2RXH2 3/20 0.54
POLB P06746 1/20 0.54
GAA P10253 1/20 0.54
LTA4H P09960 4/20 0.54
PTGS2 P35354 2/20 0.54
ATM Q13315 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
PSMB1 P20618 1/20 0.49
PSMB5 P28074 1/20 0.49
PSMB2 P49721 1/20 0.49
HRH3 Q9Y5N1 3/20 0.48
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
BACE1 P56817 1/20 0.47
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2935953 0.98 CHRNB2 (0.57) CHRNB2CHRNA4KDM4EPOLBGAA
SCHEMBL2934355 0.93 L3MBTL1 (0.56) CHRNB2CHRNA4KDM4EATML3MBTL1
SCHEMBL15884247 0.91 L3MBTL1 (0.54) CHRNB2CHRNA4KDM4EATML3MBTL1
SCHEMBL2936683 0.87 CHRNB2 (0.51) CHRNB2CHRNA4KDM4ELTA4HPTGS2
SCHEMBL3577214 0.85 TSHR (0.55) CHRNB2CHRNA4KDM4ELTA4HALDH1A1
SCHEMBL15884244 0.80 CHRNB2 (0.57) CHRNB2CHRNA4LTA4HPTGS2PSMB1
SCHEMBL18474493 0.80 CHRNB2 (0.57) CHRNB2CHRNA4KDM4ELTA4HPTGS2
SCHEMBL15884439 0.78 HRH3 (0.54) KDM4EHRH3ALDH1A1KCNH2
Hydrochloric Acid SCHEMBL7669872 0.78 CHRNB2 (0.51) CHRNB2CHRNA4GAAL3MBTL1
SCHEMBL7097968 0.77 CHRNB2 (0.66) CHRNB2CHRNA4KDM4ELTA4HPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229377-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS Wyeth LLC (US) 2010-09-22 EP disclosed
WO-2009076602-A1 5-ALKYL/ALKENYL-3-CYANOPYRIDINES AS KINASE INHIBITORS WYETH (US) 2009-06-18 WO disclosed