SCHEMBL2934284

SCHEMBL2934284

CC(C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccccc1)C(=O)O

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 2/20 0.62
CTSL P07711 5/20 0.62
CTSS P25774 2/20 0.62
CTSK P43235 2/20 0.62
PTPN1 P18031 1/20 0.56
CTSB P07858 4/20 0.56
L3MBTL1 Q9Y468 1/20 0.55
ACE P12821 2/20 0.54
GPR139 Q6DWJ6 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12516923 0.95 CTSB (0.62) PSMB5CTSLCTSSCTSKPTPN1
SCHEMBL11319330 0.88 PSMB5 (0.59) PSMB5CTSLCTSSCTSKCTSB
SCHEMBL10119250 0.86 PSMB5 (0.65) PSMB5CTSLCTSSCTSKPTPN1
SCHEMBL7318555 0.86 PSMB5 (0.65) PSMB5CTSLCTSSCTSKPTPN1
SCHEMBL11116006 0.86 CTSS (0.60) CTSSCTSK
SCHEMBL11116015 0.86 CTSS (0.60) CTSSCTSK
SCHEMBL9830316 0.85 CTSL (0.64) PSMB5CTSLCTSSCTSKCTSB
SCHEMBL9830319 0.85 CTSL (0.64) PSMB5CTSLCTSSCTSKCTSB
SCHEMBL4357736 0.84 ACE (0.68) PSMB5CTSLCTSSCTSKPTPN1
SCHEMBL4356229 0.84 ACE (0.68) PSMB5CTSLCTSSCTSKPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2229440-A2 RECOMBINANT ELASTASE PROTEINS AND METHODS OF MANUFACTURING AND USE THEREOF Proteon Therapeutics, Inc. (US) 2010-09-22 EP disclosed
WO-2009079220-A2 RECOMBINANT ELASTASE PROTEINS AND METHODS OF MANUFACTURING AND USE THEREOF PROTEON THERAPEUTICS, INC. (US) 2009-06-25 WO disclosed
US-5220029-A N-acyl derivatives of thiazolinone hydazones VITEK SYSTEMS, INC. (US) 1993-06-15 US disclosed
US-RE34284-E Contacting sample with enzyme reactive acyl thiazolinone hydrazone compound, adding oxidative coupling agents and oxidizing agents, monitoring increase in absorbance BIOMERIEUX VITEK, INC. (US) 1993-06-15 US disclosed
US-4950593-A USING THIAZOLINONE HYDRAZONE VITEK SYSTEMS, INC. (US) 1990-08-21 US disclosed
US-4308201-A SUBSTRATES; MEDICAL DIAGNOSIS TORII & CO., LTD. (JP) 1981-12-29 US disclosed