SCHEMBL2934400

SCHEMBL2934400

Nc1cc2cccoc-2c(N2CCNCC2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.40
HRH1 P35367 1/20 0.40
HRH4 Q9H3N8 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
HDAC2 Q92769 6/20 0.39
HDAC3 O15379 5/20 0.39
ABCB1 P08183 1/20 0.37
HTR1A P08908 2/20 0.36
HTR7 P34969 2/20 0.36
BRD4 O60885 1/20 0.35
ALDH1A1 P00352 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9119766 0.79 ALDH1A1 (0.37) KCNH2HRH1HRH4HRH3ABCB1
SCHEMBL2545151 0.69 HTR6 (0.47) HTR1AHTR7
SCHEMBL10078400 0.69 HRH1 (0.40) KCNH2HRH1HRH4HRH3HDAC2
SCHEMBL28869984 0.65 ADRB1 (0.48) HTR1AHTR7ALDH1A1
SCHEMBL10077099 0.64 HTR6 (0.49) HTR1AHTR7BRD4ALDH1A1BRD2
SCHEMBL5029237 0.64 ADRB1 (0.47) ALDH1A1
SCHEMBL3942886 0.62 ALDH1A1 (0.43) HRH1HRH4HRH3HTR1AHTR7
SCHEMBL28222649 0.62 HRH4 (0.44) HRH4HRH3ALDH1A1
SCHEMBL2876202 0.60 ADRB1 (0.52) KCNH2HRH1HRH4HRH3HDAC2
SCHEMBL27960523 0.59 HTR7 (0.50) HRH3HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781292-B1 EXTENDED RELEASE FORMULATION OF 3-AMINO-8-(1-PIPERAZINYL)-2H-1BENZOPYRAN-2-ONE ABBOTT HEALTHCARE PRODUCTS BV (NL) 2010-09-22 EP claimed