SCHEMBL2935441

SCHEMBL2935441

CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.55
CACNA1B Q00975 1/20 0.55
CACNA1C Q13936 1/20 0.55
TACR1 P25103 17/20 0.52
CETP P11597 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13818149 0.92 CACNA1G (0.51) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL29746466 0.92 CACNA1G (0.51) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL545966 0.90 CACNA1G (0.50) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL3005488 0.89 CACNA1G (0.49) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL25375270 0.82 CACNA1G (0.53) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL19950236 0.81 CLK1 (0.45) CACNA1GCACNA1BCACNA1C
SCHEMBL22771190 0.78 RIPK1 (0.43) CACNA1GCACNA1BCACNA1C
SCHEMBL3158285 0.78 TACR1 (0.57) TACR1
SCHEMBL12435665 0.78 TACR1 (0.57) TACR1
SCHEMBL6678261 0.77 CETP (0.43) CACNA1GCACNA1BCACNA1CTACR1CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993991-B1 PROCESS FOR THE PREPARATION OF 3,5-BIS (TRIFLUOROMETHYL)-N-METHYLBENZYLAMINE MITENI SPA (IT) 2010-09-22 EP disclosed
US-7514431-B2 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity MERCK & CO., INC. (US) 2009-04-07 US disclosed
US-7514431-B2 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity MERCK & CO., INC. (US) 2009-04-07 US disclosed
EP-1993991-A2 PROCESS FOR THE PREPARATION OF 3,5-BIS (TRIFLUOROMETHYL)-N-METHYLBENZYLAMINE MITENI S.p.A. (IT) 2008-11-26 EP disclosed
WO-2007107818-A2 PROCESS FOR THE PREPARATION OF 3,5-BIS (TRIFLUOROMETHYL)-N-METHYLBENZYLAMINE MITENI S.P.A. (IT) 2007-09-27 WO disclosed