SCHEMBL545966

SCHEMBL545966

CN(Cc1cc(N)cc(C(F)(F)F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.50
CACNA1B Q00975 1/20 0.50
CACNA1C Q13936 1/20 0.50
TACR1 P25103 16/20 0.44
CETP P11597 2/20 0.42
HTR2C P28335 1/20 0.36
SLC6A4 P31645 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2935441 0.90 CACNA1G (0.55) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL6678261 0.88 CETP (0.43) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL29746466 0.85 CACNA1G (0.51) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL13818149 0.85 CACNA1G (0.51) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL3005488 0.83 CACNA1G (0.49) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL5428175 0.82 TACR1 (0.52) TACR1
SCHEMBL10174998 0.81 RIPK1 (0.39) CACNA1GCACNA1BCACNA1CHTR2CSLC6A4
SCHEMBL25375270 0.77 CACNA1G (0.53) CACNA1GCACNA1BCACNA1CTACR1CETP
SCHEMBL2228851 0.77 HSD11B1 (0.51) HTR2CSLC6A4
SCHEMBL19950236 0.76 CLK1 (0.45) CACNA1GCACNA1BCACNA1CHTR2CSLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8110687-B2 Bicyclic compounds with kinase inhibitory activity MILLENNIUM PHARMACEUTICALS, INC. (US) 2012-02-07 US disclosed