SCHEMBL29358907

SCHEMBL29358907

COCc1ccc(C(N)=O)c(-c2ccc(Cc3cccc(Cl)c3)cn2)n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 2/20 0.42
AKT1 P31749 1/20 0.42
GPR52 Q9Y2T5 4/20 0.41
MAOB P27338 3/20 0.37
MAOA P21397 1/20 0.37
CD38 P28907 1/20 0.37
GAA P10253 1/20 0.36
S1PR4 O95977 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDE4B Q07343 1/20 0.36
GRM5 P41594 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29357073 0.88 RPS6KB1 (0.45) RPS6KB1AKT1GPR52CD38CYP11B1
SCHEMBL29355505 0.80 RPS6KB1 (0.43) RPS6KB1AKT1GPR52CD38CYP11B1
SCHEMBL29357035 0.76 RPS6KB1 (0.43) RPS6KB1AKT1GPR52MAOBCYP11B1
SCHEMBL29358277 0.75 GPR52 (0.43) RPS6KB1AKT1GPR52CYP11B1CYP11B2
SCHEMBL29358160 0.74 GPR52 (0.43) RPS6KB1AKT1GPR52CYP11B1CYP11B2
Trifluoroacetic Acid SCHEMBL29358100 0.74 RPS6KB1 (0.42) RPS6KB1AKT1GPR52CYP11B1CYP11B2
SCHEMBL29355501 0.73 GPR52 (0.41) RPS6KB1AKT1GPR52CD38CYP11B1
SCHEMBL29356932 0.73 PLA2G1B (0.41) RPS6KB1AKT1GPR52CD38GAA
SCHEMBL29355361 0.71 GPR52 (0.40) GPR52MAOBCD38CYP11B1CYP11B2
SCHEMBL21394891 0.70 ALDH1A1 (0.47) CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3941908-A1 COMPOUNDS AND USES THEREOF Yumanity Therapeutics, Inc. (US) 2022-01-26 EP disclosed